SCHEMBL7549924

SCHEMBL7549924

CN1CCNCc2cc(NC(=N)C3=CC=CCC3=S)ccc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
PKM P14618 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
THPO P40225 1/20 0.32
RAB9A P51151 1/20 0.32
HIF1A Q16665 1/20 0.32
MAPT P10636 1/20 0.32
BLM P54132 1/20 0.32
PMP22 Q01453 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
F2 P00734 1/20 0.30
PLG P00747 1/20 0.30
PLAU P00749 1/20 0.30
PLAT P00750 1/20 0.30
KLKB1 P03952 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482739 0.78 CYP1A2 (0.32) NPC1CYP1A2RAB9AMAPTSMN1; SMN2
SCHEMBL7550697 0.77 MEN1 (0.31)
SCHEMBL7554137 0.75 KDM4E (0.31) MAPT
SCHEMBL7827664 0.75 ROCK2 (0.38) CYP3A4
SCHEMBL7512695 0.74 F2 (0.31) F2PLGPLAUPLATKLKB1
SCHEMBL7549919 0.74 MAPT (0.39) NPC1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL7550546 0.74 HTR2A (0.33)
Hydrochloric Acid SCHEMBL7552145 0.74 MAPT (0.38) NPC1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL7516507 0.72 PNMT (0.42)
SCHEMBL7510864 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP claimed