SCHEMBL7516507

SCHEMBL7516507

CC1Cc2ccc(NC(=N)C3=CC=CCC3=S)cc2CN1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PNMT P11086 4/20 0.42
ADRA2A P08913 2/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
HDAC8 Q9BY41 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7506577 0.87 PNMT (0.44) PNMTADRA2AADRA2BADRA2C
SCHEMBL7511439 0.84 PNMT (0.37) PNMTADRA2AADRA2BADRA2C
SCHEMBL7512695 0.82 F2 (0.31)
SCHEMBL8305510 0.81 CA12 (0.34)
SCHEMBL7510864 0.79
SCHEMBL8307723 0.77 DRD2 (0.32)
SCHEMBL7513395 0.76 MAOA (0.39)
SCHEMBL8309882 0.75 DRD2 (0.46)
SCHEMBL7512428 0.75 L3MBTL3 (0.31)
SCHEMBL8309546 0.73 FYN (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861250-B1 AMIDINE AND ISOTHIOUREA DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2002-02-13 EP claimed