SCHEMBL7553111

SCHEMBL7553111

CCc1nc2ccccc2c(NCc2ccc(Br)cc2)c1OC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 4/20 0.47
POLB P06746 2/20 0.45
RAD52 P43351 1/20 0.45
KMT2A Q03164 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 1/20 0.43
EGFR P00533 1/20 0.42
NTRK1 P04629 1/20 0.41
ACHE P22303 2/20 0.41
HPGD P15428 1/20 0.40
GLA P06280 1/20 0.39
LMNA P02545 1/20 0.39
TSPO P30536 1/20 0.39
TOP2A P11388 1/20 0.39
BCHE P06276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27463941 0.93 APP (0.46) APPPOLBRAD52KMT2AL3MBTL1
SCHEMBL6651408 0.92 ALDH1A1 (0.48) APPPOLBRAD52KMT2AL3MBTL1
SCHEMBL7553839 0.87 APP (0.49) APPPOLBRAD52KMT2AL3MBTL1
SCHEMBL7650263 0.83 MAPT (0.53) APPPOLBRAD52KMT2AL3MBTL1
SCHEMBL6651230 0.78 APP (0.47) APPPOLBRAD52KMT2AL3MBTL1
SCHEMBL6652588 0.78 POLB (0.56) APPPOLBRAD52KMT2AL3MBTL1
SCHEMBL6655631 0.75 APP (0.44) APPPOLBRAD52KMT2AL3MBTL1
SCHEMBL7653573 0.74 APP (0.52) APPPOLBRAD52KMT2AL3MBTL1
SCHEMBL7649849 0.73 KMT2A (0.55) APPPOLBRAD52KMT2AALDH1A1
SCHEMBL7554973 0.73 APP (0.39) APPPOLBKMT2AL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218401-A1 4-BENZYLAMINOQUINOLINE CONJUGATES WITH BILE ACID AND THEIR HETEROANALOGUES, METHODS FOR PRODUCING THE SAME, MEDICAMENTS CONTAINING THESE COMPOUNDS AND THEIR USE Aventis Pharma Deutschland GmbH (DE) 2002-07-03 EP disclosed
WO-2001021642-A1 4-BENZYLAMINOQUINOLINE CONJUGATES WITH BILE ACID AND THEIR HETEROANALOGUES, METHODS FOR PRODUCING THE SAME, MEDICAMENTS CONTAINING THESE COMPOUNDS AND THEIR USE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-03-29 WO disclosed