SCHEMBL7554973

SCHEMBL7554973

Cc1nc2cccc(C)c2c(NCc2ccc(Br)cc2)c1OC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.39
CTNNB1 P35222 5/20 0.37
TCF7L2 Q9NQB0 5/20 0.37
MCHR1 Q99705 1/20 0.37
KMT2A Q03164 2/20 0.36
PPARA Q07869 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.35
ELANE P08246 1/20 0.35
CTRB1 P17538 1/20 0.35
NTRK1 P04629 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27464341 0.92 CTNNB1 (0.37) APPCTNNB1TCF7L2MCHR1KMT2A
SCHEMBL6653145 0.91 CTNNB1 (0.36) APPCTNNB1TCF7L2MCHR1KMT2A
SCHEMBL7553839 0.86 APP (0.49) APPKMT2AL3MBTL1NTRK1LMNA
SCHEMBL27464342 0.82 SMN1; SMN2 (0.41) APPCTNNB1TCF7L2MCHR1KMT2A
SCHEMBL7654278 0.82 MEN1 (0.42) APPCTNNB1TCF7L2KMT2AMEN1
SCHEMBL6651230 0.77 APP (0.47) APPKMT2AL3MBTL1MEN1NTRK1
SCHEMBL6652588 0.77 POLB (0.56) APPKMT2AL3MBTL1MEN1LMNA
SCHEMBL6655631 0.74 APP (0.44) APPKMT2AL3MBTL1NTRK1LMNA
SCHEMBL7553111 0.73 APP (0.47) APPKMT2AL3MBTL1NTRK1LMNA
SCHEMBL28054684 0.73 KDM4E (0.47) APPKMT2APPARAMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218401-A1 4-BENZYLAMINOQUINOLINE CONJUGATES WITH BILE ACID AND THEIR HETEROANALOGUES, METHODS FOR PRODUCING THE SAME, MEDICAMENTS CONTAINING THESE COMPOUNDS AND THEIR USE Aventis Pharma Deutschland GmbH (DE) 2002-07-03 EP disclosed
WO-2001021642-A1 4-BENZYLAMINOQUINOLINE CONJUGATES WITH BILE ACID AND THEIR HETEROANALOGUES, METHODS FOR PRODUCING THE SAME, MEDICAMENTS CONTAINING THESE COMPOUNDS AND THEIR USE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-03-29 WO disclosed