SCHEMBL7553195

SCHEMBL7553195

CC(C/C=C\c1cccc(F)c1)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.40
PTGS1 P23219 2/20 0.38
PTGS2 P35354 1/20 0.38
NFE2L2 Q16236 6/20 0.38
NR1H4 Q96RI1 2/20 0.37
RELA Q04206 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
HPGD P15428 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
EPOR P19235 1/20 0.35
AAK1 Q2M2I8 1/20 0.35
APP P05067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550965 1.00 PIN1 (0.40) PIN1PTGS1PTGS2NFE2L2NR1H4
SCHEMBL7550970 1.00 PIN1 (0.40) PIN1PTGS1PTGS2NFE2L2NR1H4
SCHEMBL7547697 0.81 GRIK1 (0.45) PTGS2AAK1
SCHEMBL7554007 0.81 GRIK1 (0.45) PTGS2AAK1
SCHEMBL7547700 0.81 GRIK1 (0.45) PTGS2AAK1
SCHEMBL3325118 0.80 CHRNB2 (0.49) PTGS1PTGS2NFE2L2
SCHEMBL3325125 0.80 CHRNB2 (0.49) PTGS1PTGS2NFE2L2
SCHEMBL7549401 0.79 AAK1 (0.41) NR1H4AAK1
SCHEMBL7549408 0.79 AAK1 (0.41) NR1H4AAK1
SCHEMBL3322749 0.78 MMP13 (0.34) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214288-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE Targacept Inc. (US) 2002-06-19 EP disclosed
WO-2001017943-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE TARGACEPT, INC. (US) 2001-03-15 WO disclosed