SCHEMBL7555860

SCHEMBL7555860

COc1ccc(CN2Cc3sc(NC4CCCCO4)c(C(=O)O)c3CC2CNC(=O)Cc2c(C)[nH]c3ccc(OC)cc23)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 1/20 0.37
PTPN5 P54829 1/20 0.36
MTNR1A P48039 3/20 0.36
MTNR1B P49286 3/20 0.36
KDM4E B2RXH2 4/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
RECQL P46063 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GAA P10253 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
HDAC1 Q13547 5/20 0.33
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
NPC1 O15118 1/20 0.32
HDAC3 O15379 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5837745 0.87 PTPN1 (0.44) AKR1C2PTPN5MTNR1AMTNR1BKDM4E
SCHEMBL7550192 0.84 AKR1C2 (0.38) AKR1C2PTPN5MTNR1AMTNR1BKDM4E
SCHEMBL7699895 0.82 KMT2A (0.42) MTNR1AMTNR1BKDM4EMEN1KMT2A
SCHEMBL7702706 0.80 KDM4E (0.41) KDM4ELMNAMEN1KMT2ACYP2C9
SCHEMBL5838311 0.80 AKR1C2 (0.39) AKR1C2PTPN5MTNR1AMTNR1BKDM4E
SCHEMBL5837754 0.79 AKR1C2 (0.36) AKR1C2PTPN5MTNR1AMTNR1BKDM4E
SCHEMBL7701621 0.77 HDAC1 (0.36) KDM4ELMNAKMT2ACYP2C9CYP2C19
SCHEMBL7542021 0.77 PTPN1 (0.38) GAAMEN1KMT2A
SCHEMBL7694698 0.77 BCHE (0.40) KDM4ELMNAPOLBMEN1KMT2A
SCHEMBL7571116 0.76 ALDH1A1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214324-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK A/S (DK) 2002-06-19 EP claimed
WO-2001019830-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) NOVO NORDISK A/S (DK) 2001-03-22 WO claimed