SCHEMBL7556199

SCHEMBL7556199

O=C(NCC[C]1CCCCCCC1)c1cc(CN2CCNCC2)ccc1Cl.[CH2].[CH2]

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.62
CHRM3 P20309 3/20 0.51
GAA P10253 1/20 0.45
MCHR1 Q99705 4/20 0.44
PAICS P22234 1/20 0.42
CYP2D6 P10635 1/20 0.42
CHRM1 P11229 1/20 0.42
HTR2A P28223 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3951445 0.89 P2RX7 (0.64) P2RX7CHRM3GAAPAICS
SCHEMBL7661977 0.87 P2RX7 (0.61) P2RX7CHRM3GAACHRM1
SCHEMBL7516797 0.80 CYP4F2 (0.44) P2RX7GAA
SCHEMBL7660243 0.79 P2RX7 (0.82) P2RX7CHRM3
SCHEMBL7663299 0.76 P2RX7 (1.00) P2RX7
SCHEMBL7657585 0.75 P2RX7 (0.93) P2RX7
SCHEMBL7559952 0.73 P2RX7 (0.61) P2RX7CHRM3CYP2D6HTR2A
SCHEMBL5142841 0.71 NPC1 (0.44) P2RX7
SCHEMBL7553515 0.71 P2RX7 (0.58) P2RX7CHRM3CYP2D6HTR2A
SCHEMBL7555457 0.70 P2RX7 (0.47) P2RX7CHRM3CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171432-A1 ADAMANTANE DERIVATIVES AstraZeneca AB (SE) 2002-01-16 EP disclosed
WO-2000061569-A1 ADAMANTANE DERIVATIVES ASTRAZENECA AB (SE) 2000-10-19 WO disclosed