Bicarbonate

Bicarbonate

SCHEMBL7556709

FC(F)(F)C1CCCCC1.O=C(O)O

nearest known ligand 0.38

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
EPHX1 P07099 7/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP3A4 P08684 1/20 0.33
EPHX2 P34913 1/20 0.33
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
SSTR4 P31391 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27490624 0.86 RXFP1 (0.34) CES2CES1KEAP1NFE2L2PDK1
SCHEMBL59958 0.86 NOS3 (0.32) ALDH1A1
SCHEMBL22068846 0.86 NOS3 (0.32) ALDH1A1
SCHEMBL18643888 0.86 NOS3 (0.32) ALDH1A1
Methyl Alcohol SCHEMBL28003807 0.83 PDK1 (0.33) PDK1PDK2PDK3PDK4EPHX1
Ammonia Solution, Strong SCHEMBL18669725 0.83 NOS3 (0.31)
SCHEMBL15641746 0.83 NOS3 (0.33) ALDH1A1
SCHEMBL15184 0.83
SCHEMBL9000709 0.77 KEAP1 (0.39) CES2CES1KEAP1NFE2L2PDK1
SCHEMBL554737 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1220841-A2 TRIFLUOROMETHYL-SUBSTITUTED SPIROCYCLIC KETOENOLS Bayer Aktiengesellschaft (DE) 2002-07-10 EP disclosed
WO-2001023354-A2 TRIFLUOROMETHYL-SUBSTITUTED SPIROCYCLIC KETOENOLS AND USE THEREOF AS PESTICIDES AND HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2001-04-05 WO disclosed
EP-0418362-B1 TRIFLUOROMETHYLCYCLOHEXANE DERIVATIVES MERCK PATENT GMBH (DE) 1995-01-04 EP disclosed
EP-0418362-A1 TRIFLUOROMETHYLCYCLOHEXANE DERIVATIVES. MERCK PATENT GMBH (DE) 1991-03-27 EP disclosed
WO-1990012073-A1 TRIFLUOROMETHYLCYCLOHEXANE DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1990-10-18 WO disclosed
EP-0300218-A1 Use of substituted 1,4-naphthoquinones against nites and fungi BAYER AG (DE) 1989-01-25 EP disclosed