SCHEMBL7558580

SCHEMBL7558580

COc1cccc(NC(=O)NC2=CC(=O)NC2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.59
TSHR P16473 1/20 0.59
ALDH1A1 P00352 3/20 0.59
KDR P35968 1/20 0.56
RAB9A P51151 12/20 0.55
NPC1 O15118 10/20 0.55
MITF O75030 1/20 0.55
CASP3 P42574 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
MAPT P10636 8/20 0.53
SMN1; SMN2 Q16637 6/20 0.53
KMT2A Q03164 6/20 0.53
HTT P42858 5/20 0.53
MEN1 O00255 5/20 0.53
LMNA P02545 2/20 0.53
MAPK1 P28482 1/20 0.53
STAT1 P42224 1/20 0.53
RAF1 P04049 1/20 0.53
GAA P10253 2/20 0.52
USP2 O75604 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31040569 0.81 TP53 (0.87) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL4893387 0.81 TP53 (0.87) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL17084260 0.79 TP53 (0.84) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL7523675 0.78 RAB9A (0.59) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL7525489 0.78 TP53 (0.59) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL14442613 0.76 TP53 (0.84) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL29556598 0.74 TP53 (0.70) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL22103808 0.74 TP53 (0.74) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL6388689 0.73 TP53 (0.73) TP53TSHRALDH1A1RAB9ANPC1
SCHEMBL7610775 0.73 TP53 (0.73) TP53TSHRALDH1A1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173420-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY Novuspharma S.p.A. (IT) 2002-01-23 EP disclosed
WO-2000053581-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY NOVUSPHARMA S.P.A. (IT) 2000-09-14 WO disclosed