SCHEMBL7558640

SCHEMBL7558640

COc1ccc(-c2noc(C)c2C(N)=O)cc1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.68
GAA P10253 2/20 0.68
KMT2A Q03164 2/20 0.68
GPBAR1 Q8TDU6 1/20 0.59
PTGS2 P35354 1/20 0.59
BACE1 P56817 7/20 0.57
TSHR P16473 2/20 0.54
LMNA P02545 2/20 0.53
TP53 P04637 1/20 0.53
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
KDM4E B2RXH2 1/20 0.52
ALOX12 P18054 1/20 0.52
HTT P42858 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
HSD17B10 Q99714 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2777180 0.87 PTGS2 (0.60) MEN1GAAKMT2AGPBAR1PTGS2
SCHEMBL11893877 0.85 ALDH1A1 (0.61) MEN1GAAKMT2AGPBAR1PTGS2
SCHEMBL2723582 0.85 GPBAR1 (0.62) MEN1GAAKMT2AGPBAR1PTGS2
SCHEMBL11411843 0.83 LMNA (0.61) MEN1GAAKMT2AGPBAR1PTGS2
SCHEMBL4718673 0.82 KMT2A (0.72) MEN1GAAKMT2AGPBAR1PTGS2
SCHEMBL2775071 0.82 GAA (0.64) GAAGPBAR1PTGS2BACE1TSHR
SCHEMBL903110 0.81 KMT2A (1.00) MEN1GAAKMT2ATSHRALDH1A1
Hydrochloric Acid SCHEMBL30684627 0.81 KMT2A (0.70) MEN1GAAKMT2AGPBAR1PTGS2
Hydrochloric Acid SCHEMBL30684473 0.80 KMT2A (0.97) MEN1GAAKMT2ATSHRALDH1A1
Hydrochloric Acid SCHEMBL30684542 0.80 KMT2A (0.97) MEN1GAAKMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1226131-A2 ISOXAZOLECARBOXAMIDE DERIVATIVES RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.p.a. (IT) 2002-07-31 EP claimed
WO-2001029015-A2 ISOXAZOLECARBOXAMIDE DERIVATIVES AS ALPHA1-ADRENERGIC RECEPTOR ANTAGONISTS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.P.A. (IT) 2001-04-26 WO claimed