SCHEMBL7560104

SCHEMBL7560104

O=C(N[CH]c1ccccc1)NN1CCOCC1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 5/20 0.47
CDK5R1 Q15078 5/20 0.47
CCNA2 P20248 3/20 0.47
CDK2 P24941 3/20 0.47
CCNA1 P78396 3/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
CYP2D6 P10635 1/20 0.43
POLB P06746 2/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
LIPE Q05469 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL219620 0.76 SMN1; SMN2 (0.67) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL7562512 0.75 POLB (0.65) SMN1; SMN2POLBGAAMAPTMEN1
SCHEMBL7660168 0.74 RAB9A (0.58) RAB9ASMN1; SMN2NPC1POLBMAPT
SCHEMBL3955220 0.72 SMN1; SMN2 (0.71) SMN1; SMN2CYP2D6POLBGAAMAPT
SCHEMBL6790329 0.72 SMN1; SMN2 (0.59) CDK5CDK5R1RAB9ASMN1; SMN2NPC1
SCHEMBL7660162 0.71 LMNA (0.50) RAB9ASMN1; SMN2CYP2D6POLBGAA
SCHEMBL11668271 0.71 SMN1; SMN2 (0.56) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL7298618 0.71 KMT2A (0.58) CDK5CDK5R1CCNA2CDK2CCNA1
SCHEMBL14096485 0.70 KMT2A (0.66) RAB9ANPC1POLBGAAMAPT
SCHEMBL10757188 0.69 LIPE (0.73) RAB9ASMN1; SMN2NPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002067654-A3 6-SUBSTITUTED PYRAZOLO[3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-10-31 WO claimed
WO-2002067654-A3 6-SUBSTITUTED PYRAZOLO[3,4-D]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2002-10-31 WO disclosed
EP-1121363-A2 6-SUBSTITUTED PYRAZOLO 3,4-d]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS Du Pont Pharmaceuticals Company (US) 2001-08-08 EP disclosed
WO-2000021926-A2 6-SUBSTITUTED PYRAZOLO[3,4-d]PYRIMIDIN-4-ONES USEFUL AS CYCLIN DEPENDENT KINASE INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 2000-04-20 WO disclosed