SCHEMBL756324

SCHEMBL756324

CC(C)(N)c1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.50
CYP2A6 P11509 1/20 0.44
CA2 P00918 2/20 0.41
CA1 P00915 1/20 0.41
CA5A P35218 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 2/20 0.41
ALOX15 P16050 2/20 0.41
MAPK1 P28482 1/20 0.41
AKT1 P31749 1/20 0.39
AKT2 P31751 1/20 0.39
NOS1 P29475 2/20 0.36
OGG1 O15527 1/20 0.34
CDK1 P06493 1/20 0.34
KDR P35968 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
HTT P42858 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL992228 0.97 PDE2A (0.48) PDE2ACYP2A6CA2CA1CA5A
Iodide SCHEMBL25233569 0.97 PDE2A (0.48) PDE2ACYP2A6CA2CA1CA5A
SCHEMBL1706121 0.85 PDE2A (0.62) PDE2AALDH1A1ALOX15MAPK1AKT1
SCHEMBL27985809 0.79 CA1 (0.48) PDE2ACYP2A6CA2CA1CA5A
SCHEMBL7944567 0.79 CYP2A6 (0.40) CYP2A6CA2CA1CA5ACA9
SCHEMBL3979356 0.79 CYP2A6 (0.40) PDE2ACYP2A6CA2CA1CA5A
SCHEMBL16887733 0.79 CYP2A6 (0.40) PDE2ACYP2A6CA2CA1CA5A
SCHEMBL1025732 0.79 CYP2A6 (0.40) PDE2ACYP2A6CA2CA1CA5A
SCHEMBL18548321 0.78 CYP2A6 (0.44) CYP2A6CA2CA1CA5ACA9
SCHEMBL5080121 0.77 CYP2A6 (0.50) PDE2ACYP2A6CA2CA1CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 310 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019367-A1 DERIVATIVES OF 2,5- AND 3,5-DISUBSTITUTED ANILINES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2000-07-19 EP claimed
WO-1999007672-A1 DERIVATIVES OF 2,5- AND 3,5-DISUBSTITUTED ANILINES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1999-02-18 WO claimed
US-12552771-B2 Carboxylic acid containing azetidinyl compounds for the treatment of neurodegenerative diseases CELGENE CORPORATION (US) 2026-02-17 US disclosed
EP-4306529-B1 FGFR INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS INC (US) 2026-01-21 EP disclosed
US-12527776-B2 Treatment of ciliopathies using inhibitors of glucosylceramide synthase (GCS) GENZYME CORPORATION (US) 2026-01-20 US disclosed
US-12522605-B2 FGFR inhibitors and methods of use thereof RELAY THERAPEUTICS, INC. (US) 2026-01-13 US disclosed
US-12509424-B2 Compound and composition as PDGF receptor kinase inhibitor NIPPON SHINYAKU CO., LTD. (JP) 2025-12-30 US disclosed
EP-4651872-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE TO TREAT HYPOPARATHYROIDISM AND OSTEOPOROSIS Septerna, Inc. (US) 2025-11-26 EP disclosed
EP-4021901-B1 SUBSTITUTED PYRIDOPYRIMIDINONYL COMPOUNDS USEFUL AS T CELL ACTIVATORS BRISTOL MYERS SQUIBB CO (US) 2025-09-24 EP disclosed
US-12378224-B2 Heteroaryl compounds and their use as Mer inhibitors DONG-A SOCIO HOLDINGS CO., LTD. (KR) 2025-08-05 US disclosed
US-20250205219-A1 TARGETED DEGRADATION OF VAV1 MONTE ROSA THERAPEUTICS AG (CH) 2025-06-26 US disclosed
EP-1222175-A1 4,5-DISUBSTITUTED-2-AMINOPYRIMIDINES Celltech R&D Limited (GB) 2002-07-17 EP disclosed
WO-2001029009-A1 4,5-DISUBSTITUTED-2-AMINOPYRIMIDINES CELLTECH R&D LIMITED (GB) 2001-04-26 WO disclosed
EP-1019367-A1 DERIVATIVES OF 2,5- AND 3,5-DISUBSTITUTED ANILINES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2000-07-19 EP disclosed
CN-1051299-C Tetrahydrophthamide derivative medium for preparation of same, preparation of same and herbcide which uses same as effective composition SAGAMI CHEM RES (JP) 2000-04-12 CN disclosed
WO-1999007672-A1 DERIVATIVES OF 2,5- AND 3,5-DISUBSTITUTED ANILINES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1999-02-18 WO disclosed
EP-0635485-B1 TETRAHYDROPHTHALAMIDE DERIVATIVE, INTERMEDIATE FOR PRODUCING THE SAME, PRODUCTION OF BOTH, AND HERBICIDE CONTAINING THE SAME AS ACTIVE INGREDIENT SAGAMI CHEM RES (JP) 1997-06-11 EP disclosed
US-5506190-A Tetrahydrophthalamide derivative, intermediate for producing the same, production of both, and herbicide containing the same as active ingredient SAGAMI CHEMICAL RESEARCH CENTER (JP) 1996-04-09 US disclosed
EP-0635485-A1 TETRAHYDROPHTHALAMIDE DERIVATIVE, INTERMEDIATE FOR PRODUCING THE SAME, PRODUCTION OF BOTH, AND HERBICIDE CONTAINING THE SAME AS ACTIVE INGREDIENT SAGAMI CHEMICAL RESEARCH CENTER (JP) 1995-01-25 EP disclosed
CN-1084847-A Tetrahydrochysene butyl benzene orthobenzol diacid amide derivative and its preparation intermediate and manufacture method thereof and with its weedicide as effective constituent SAGAMI CHEM RES (JP) 1994-04-06 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12527776-B2 Treatment of ciliopathies using inhibitors of glucosylceramide synthase (GCS) GBA1, GBA2, GALC PDE2A 1821/4885CYP2A6 2075/4885CA2 4155/4885
US-12378224-B2 Heteroaryl compounds and their use as Mer inhibitors MERTK, RET, ERBB2 PDE2A 3902/4885CYP2A6 1320/4885CA2 3399/4885
US-12509424-B2 Compound and composition as PDGF receptor kinase inhibitor PDGFRA, PDGFRB, PDGFA PDE2A 1013/4885CYP2A6 3817/4885CA2 339/4885
US-20250205219-A1 TARGETED DEGRADATION OF VAV1 VAV1, KRAS, CBL PDE2A 2926/4885CYP2A6 4589/4885CA2 4034/4885
US-12552771-B2 Carboxylic acid containing azetidinyl compounds for the treatment of neurodegenerative diseases S1PR5, CLN6, SNCA PDE2A 1013/4885CYP2A6 282/4885CA2 325/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.