SCHEMBL8167993

SCHEMBL8167993

COc1ccc(CC[N+](C)(C)C[C@@H](O)COc2ccc(N(C)S(=O)(=O)c3ccc(C)cc3)cc2C#N)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
MAPT P10636 3/20 0.46
LMNA P02545 3/20 0.46
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRB2 P07550 1/20 0.37
CYP2D6 P10635 1/20 0.37
ADRB3 P13945 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
CASR P41180 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KCNH2 Q12809 1/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8165088 0.88 ADRB3 (0.40) ALDH1A1MEN1KMT2AADRB2CYP2D6
SCHEMBL8166640 0.88 ALDH1A1 (0.53) ALDH1A1LMNAKEAP1NFE2L2KMT2A
Hydrochloric Acid SCHEMBL8159978 0.88 SLC6A2 (0.40) ALDH1A1MEN1KMT2AADRB2CYP2D6
SCHEMBL8169018 0.83 ADRB2 (0.47) ALDH1A1MAPTADRB2ADRB3
SCHEMBL6862114 0.82 CASR (0.61) ALDH1A1ADRB2CYP2D6ADRB3SLC6A2
SCHEMBL6862107 0.82 CASR (0.61) ALDH1A1ADRB2CYP2D6ADRB3SLC6A2
Hydrochloric Acid SCHEMBL7802320 0.82 CASR (0.60) ALDH1A1ADRB2CYP2D6ADRB3SLC6A2
Hydrochloric Acid SCHEMBL6863037 0.82 CASR (0.60) ALDH1A1ADRB2CYP2D6ADRB3SLC6A2
SCHEMBL7563669 0.81 CASR (0.48) ALDH1A1KEAP1NFE2L2ADRB2CYP2D6
SCHEMBL8169408 0.80 KEAP1 (0.45) ALDH1A1MAPTLMNAKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-01-26 EP disclosed
WO-1998045255-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-15 WO disclosed