SCHEMBL7563875

SCHEMBL7563875

COc1cccc(CNc2ccc(C(C)=O)cc2)c1OCCCC(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.61
MEN1 O00255 1/20 0.61
SMN1; SMN2 Q16637 4/20 0.60
HIF1A Q16665 3/20 0.55
NPC1 O15118 3/20 0.50
RAB9A P51151 2/20 0.50
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
HTT P42858 2/20 0.50
HSP90AA1 P07900 1/20 0.50
HPGD P15428 1/20 0.50
LMNA P02545 4/20 0.47
NPSR1 Q6W5P4 2/20 0.47
FFAR4 Q5NUL3 2/20 0.47
MAPT P10636 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
TP53 P04637 1/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7567727 0.78 ALOX12 (0.60) KMT2AMEN1SMN1; SMN2HIF1ANPC1
SCHEMBL4820844 0.71 HIF1A (0.72) KMT2AMEN1SMN1; SMN2HIF1ANPC1
SCHEMBL7563849 0.70 POLB (0.51) KMT2ASMN1; SMN2ALDH1A1HPGDLMNA
SCHEMBL8078072 0.69 PPARA (0.53) SMN1; SMN2LMNAFFAR4
SCHEMBL3697457 0.69 LMNA (0.50) SMN1; SMN2ALDH1A1LMNAFFAR4L3MBTL1
SCHEMBL15613891 0.68 HSD17B10 (0.57) SMN1; SMN2NPC1RAB9AALDH1A1MAPT
SCHEMBL2553169 0.68 KMT2A (0.63) KMT2AMEN1SMN1; SMN2ALDH1A1HTT
SCHEMBL28134005 0.68 ALDH1A1 (0.61) KMT2AMEN1SMN1; SMN2HIF1ANPC1
SCHEMBL612449 0.68 FFAR4 (0.51) KMT2AMEN1HIF1AKDM4EALDH1A1
SCHEMBL7086937 0.67 LMNA (0.51) KMT2AMEN1ALDH1A1LMNAFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0689845-B1 Conjugates of methyltrithio antitumor agents and intermediates for their synthesis AMERICAN CYANAMID CO (US) 2002-09-04 EP disclosed
US-5773001-A ANTIGROWTH AGENTS AMERICAN CYANAMID COMPANY (US) 1998-06-30 US disclosed
EP-0689845-A2 Conjugates of methyltrithio antitumor agents and intermediates for their synthesis AMERICAN CYANAMID COMPANY (US) 1996-01-03 EP disclosed