SCHEMBL7565119

SCHEMBL7565119

CCOC(=O)C[C@H](NC(=O)CC(=O)NCCCC1=CC=C2CCCNC2N1)c1cccnc1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.34
ITGB3 P05106 16/20 0.34
ITGAV P06756 10/20 0.34
KCNA5 P22460 1/20 0.34
ITGA2B P08514 7/20 0.34
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7571407 0.90 ITGB3 (0.43) ITGB3ITGAVITGA2B
SCHEMBL7587023 0.80 TSHR (0.34)
SCHEMBL7009188 0.77 ITGB3 (0.57) ITGB3ITGAVITGA2B
SCHEMBL7009184 0.77 ITGB3 (0.57) ITGB3ITGAVITGA2B
SCHEMBL7565113 0.71 ROCK2 (0.34) ROCK2ITGB3ITGAVKCNA5ITGA2B
SCHEMBL7552889 0.71 ITGAV (0.45) ITGB3ITGAVITGA2B
SCHEMBL7590655 0.71 ITGAV (0.45) ITGB3ITGAVITGA2B
SCHEMBL7592208 0.71 ITGAV (0.45) ITGB3ITGAVITGA2B
SCHEMBL7373638 0.68 ITGB3 (0.44) ROCK2ITGB3ITGAVKCNA5ITGA2B
SCHEMBL6739002 0.68 ITGB3 (0.44) ROCK2ITGB3ITGAVKCNA5ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946165-A4 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2001-04-11 EP claimed
EP-0946165-A1 INTEGRIN ANTAGONISTS Merck & Co., Inc. (US) 1999-10-06 EP claimed
WO-1998018460-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-05-07 WO claimed
EP-0946165-A4 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2001-04-11 EP disclosed
EP-0946165-A1 INTEGRIN ANTAGONISTS Merck & Co., Inc. (US) 1999-10-06 EP disclosed
WO-1998018460-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-05-07 WO disclosed