SCHEMBL7571407

SCHEMBL7571407

O=C(O)C[C@H](NC(=O)CC(=O)NCCCC1=CC=C2CCCNC2N1)c1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.43
ITGAV P06756 15/20 0.43
ITGA2B P08514 7/20 0.42
ITGB5 P18084 1/20 0.39
ITGB6 P18564 1/20 0.39
ITGB8 P26012 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7565119 0.90 ROCK2 (0.34) ITGB3ITGAVITGA2B
SCHEMBL7590655 0.80 ITGAV (0.45) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7592208 0.80 ITGAV (0.45) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7552889 0.80 ITGAV (0.45) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7008303 0.75 ITGB3 (0.70) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7008295 0.75 ITGB3 (0.70) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7591261 0.74 ITGAV (0.61) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7589125 0.74 ITGAV (0.61) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7575089 0.73 ITGB3 (0.62) ITGB3ITGAVITGA2BITGB5ITGB6
SCHEMBL7552205 0.71 ITGAV (0.41) ITGB3ITGAVITGB5ITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946165-A4 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2001-04-11 EP disclosed
EP-0946165-A1 INTEGRIN ANTAGONISTS Merck & Co., Inc. (US) 1999-10-06 EP disclosed
WO-1998018460-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-05-07 WO disclosed