SCHEMBL7565495

SCHEMBL7565495

CC(=O)c1ccc2c(c1)N(CCCCCCO)c1ccccc1S2

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.74
HTR1A P08908 4/20 0.74
DRD2 P14416 4/20 0.74
SLC6A2 P23975 4/20 0.74
SLC6A4 P31645 4/20 0.74
ADRA1A P35348 4/20 0.74
DRD3 P35462 4/20 0.74
SLC6A3 Q01959 4/20 0.74
KCNH2 Q12809 4/20 0.74
ADRA2A P08913 3/20 0.74
ADRA2B P18089 3/20 0.74
ADRA2C P18825 3/20 0.74
HTR2A P28223 3/20 0.74
HTR2B P41595 3/20 0.74
DRD1 P21728 2/20 0.74
MLNR O43193 1/20 0.74
ESR1 P03372 1/20 0.74
PTGS2 P35354 1/20 0.74
HRH3 Q9Y5N1 1/20 0.74
CYP1A2 P05177 4/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24439565 0.95 HRH1 (0.77) HRH1HTR1ADRD2SLC6A2SLC6A4
SCHEMBL9475738 0.90 HTR1A (0.77) HRH1HTR1ADRD2SLC6A2SLC6A4
SCHEMBL7566877 0.88 HTR1A (0.70) HRH1HTR1ADRD2SLC6A2SLC6A4
SCHEMBL4730313 0.88 HTR1A (0.76) HRH1HTR1ADRD2SLC6A2SLC6A4
SCHEMBL29062451 0.86 HTR1A (0.74) HRH1HTR1ADRD2SLC6A2SLC6A4
SCHEMBL9380936 0.86 HTR1A (0.74) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL94266 0.85 HRH1 (1.00) HRH1HTR1ADRD2SLC6A2SLC6A4
Acetophenazine SCHEMBL29710923 0.85 HRH1 (1.00) HRH1HTR1ADRD2SLC6A2SLC6A4
Acepromazine SCHEMBL73018 0.84 CYP2D6 (1.00) HRH1HTR1ADRD2SLC6A2SLC6A4
Acepromazine SCHEMBL29582179 0.84 CYP2D6 (1.00) HRH1HTR1ADRD2SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0689845-B1 Conjugates of methyltrithio antitumor agents and intermediates for their synthesis AMERICAN CYANAMID CO (US) 2002-09-04 EP disclosed
EP-0689845-A2 Conjugates of methyltrithio antitumor agents and intermediates for their synthesis AMERICAN CYANAMID COMPANY (US) 1996-01-03 EP disclosed