SCHEMBL7565538

SCHEMBL7565538

C=C1C(c2ccccc2)=C(c2cc(C)cs2)C1(Cl)Cl

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6326345 0.83 PTGS1 (0.34) PTGS1PTGS2
SCHEMBL7568017 0.72 PTGS1 (0.47) PTGS1PTGS2
SCHEMBL72613 0.72 AR (0.43)
SCHEMBL7567949 0.71 PTGS1 (0.44) PTGS1PTGS2
SCHEMBL7569141 0.69 PTGS1 (0.37) PTGS1PTGS2
SCHEMBL7565479 0.69 PTGS2 (0.35) PTGS1PTGS2
SCHEMBL7573867 0.67 PTGS1 (0.47) PTGS1PTGS2
SCHEMBL7565527 0.66 PTGS2 (0.51) PTGS1PTGS2
SCHEMBL7566050 0.66 ALDH2 (0.32)
SCHEMBL10472855 0.65 HSD17B1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889878-B1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC (CA) 2002-09-04 EP disclosed
EP-0889878-A1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC. (CA) 1999-01-13 EP disclosed
US-5817700-A ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1998-10-06 US disclosed
WO-1997036863-A1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC. (CA) 1997-10-09 WO disclosed