SCHEMBL7567949

SCHEMBL7567949

C=C1CC(c2cc(C)cs2)=C1c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
AR P10275 1/20 0.31
SLC6A7 Q99884 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7566081 0.82 PTGS1 (0.46) PTGS1PTGS2ARSLC6A7
SCHEMBL7567903 0.76 PTGS2 (0.34) PTGS1PTGS2NPC1HPGDTSHR
SCHEMBL7569459 0.75 HDAC1 (0.34) SLC6A7
SCHEMBL5833325 0.75 KMT2A (0.56) PTGS1PTGS2SMN1; SMN2
SCHEMBL72613 0.74 AR (0.43) NPC1HPGDTSHRRAB9ASMN1; SMN2
SCHEMBL7565538 0.71 PTGS1 (0.33) PTGS1PTGS2
SCHEMBL8609716 0.70 HPGD (0.36) NPC1HPGDRAB9ASMN1; SMN2
SCHEMBL10472855 0.67 HSD17B1 (0.47) NPC1HPGDRAB9ASMN1; SMN2
SCHEMBL7568017 0.66 PTGS1 (0.47) PTGS1PTGS2NPC1TSHRRAB9A
SCHEMBL7566050 0.65 ALDH2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889878-B1 BISARYLCYCLOBUTENE DERIVATES AS CYCLOOXYGENASE INHIBITORS MERCK FROSST CANADA INC (CA) 2002-09-04 EP disclosed
US-5817700-A ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1998-10-06 US disclosed