SCHEMBL7567314

SCHEMBL7567314

COC(=O)c1ccc(NS(=O)(=O)c2cccc(C(F)(F)F)c2)c(NS(=O)(=O)c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.59
GAA P10253 2/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
SLC20A2 Q08357 1/20 0.52
SLC20A1 Q8WUM9 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
MMP1 P03956 1/20 0.52
MMP2 P08253 1/20 0.52
MMP9 P14780 1/20 0.52
MMP8 P22894 1/20 0.52
MMP13 P45452 1/20 0.52
ACLY P53396 3/20 0.52
CYP2C9 P11712 3/20 0.50
HSD17B2 P37059 1/20 0.50
SLC40A1 Q9NP59 2/20 0.49
CCR2 P41597 1/20 0.49
LMNA P02545 1/20 0.49
ALDH1A1 P00352 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7570517 0.94 CYP2C9 (0.61) NPSR1GAAMEN1KMT2ASLC20A2
SCHEMBL7578595 0.90 NPSR1 (0.72) NPSR1GAAMEN1KMT2ASLC20A2
SCHEMBL7572555 0.86 CYP2C9 (0.60) NPSR1MEN1KMT2AACLYCYP2C9
SCHEMBL19065100 0.84 GAA (0.64) GAAMEN1KMT2ACA1CA2
SCHEMBL7569668 0.82 KMT2A (0.76) NPSR1GAAMEN1KMT2ASLC20A2
SCHEMBL7572438 0.81 SLC20A2 (0.63) NPSR1GAAMEN1KMT2ASLC20A2
SCHEMBL23022352 0.81 CYP2C9 (0.57) NPSR1GAAMEN1KMT2AACLY
SCHEMBL7572561 0.80 NPSR1 (0.66) NPSR1GAAMEN1KMT2ASLC20A2
SCHEMBL22498190 0.80 CACNA1B (0.56) NPSR1GAAMEN1KMT2ACA1
SCHEMBL29528521 0.80 CACNA1B (0.56) NPSR1GAAMEN1KMT2ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002083629-A1 BISSULFONAMIDE DERIVATIVES AS INHIBITORS OF DEHYDROQUINATE SYNTHETASES AND TYPE II DEHYDROQUINASES ARROW THERAPEUTICS LIMITED (GB) 2002-10-24 WO disclosed
EP-1239852-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS Arrow Therapeutics Limited (GB) 2002-09-18 EP disclosed
WO-2001028537-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS ARROW THERAPEUTICS LIMITED (GB) 2001-04-26 WO disclosed