SCHEMBL7570517

SCHEMBL7570517

COC(=O)c1ccc(NS(=O)(=O)c2cccc(C(F)(F)F)c2)c(NS(=O)(=O)c2ccc(C)cc2)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.61
NPSR1 Q6W5P4 3/20 0.56
TCF4 P15884 1/20 0.56
CTNNB1 P35222 1/20 0.56
FFAR4 Q5NUL3 2/20 0.55
FFAR1 O14842 1/20 0.55
CDK1 P06493 1/20 0.55
CCNB1 P14635 1/20 0.55
CCNA2 P20248 1/20 0.55
CDK2 P24941 1/20 0.55
CDK7 P50613 1/20 0.55
CCNH P51946 1/20 0.55
CCNA1 P78396 1/20 0.55
ALDH1A1 P00352 4/20 0.53
LMNA P02545 2/20 0.53
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
POLB P06746 2/20 0.52
TP53 P04637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7567314 0.94 NPSR1 (0.59) CYP2C9NPSR1ALDH1A1LMNAMEN1
SCHEMBL7578595 0.86 NPSR1 (0.72) NPSR1ALDH1A1LMNAKDM4EMEN1
SCHEMBL7572555 0.85 CYP2C9 (0.60) CYP2C9NPSR1ALDH1A1LMNAKDM4E
SCHEMBL7571635 0.85 FFAR1 (0.66) NPSR1FFAR4FFAR1CDK1CCNB1
SCHEMBL7573928 0.85 CYP2C9 (0.82) CYP2C9NPSR1TCF4CTNNB1FFAR4
SCHEMBL7572541 0.82 FFAR1 (0.62) NPSR1FFAR4FFAR1CDK1CCNB1
SCHEMBL7572374 0.79 NPSR1 (0.58) CYP2C9NPSR1ALDH1A1LMNAKDM4E
SCHEMBL19065100 0.79 GAA (0.64) TCF4CTNNB1FFAR4FFAR1CDK1
SCHEMBL3528690 0.79 KDM1A (0.61) CYP2C9NPSR1FFAR4FFAR1CDK1
SCHEMBL23022352 0.78 CYP2C9 (0.57) CYP2C9NPSR1TCF4CTNNB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1239852-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS Arrow Therapeutics Limited (GB) 2002-09-18 EP disclosed
WO-2001028537-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS ARROW THERAPEUTICS LIMITED (GB) 2001-04-26 WO disclosed