SCHEMBL7569359

SCHEMBL7569359

O=C(O)c1cccc2cc3cc(-c4ccccc4)ccc3nc12

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
DHODH Q02127 8/20 0.50
PARP1 P09874 1/20 0.49
ACMSD Q8TDX5 4/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
HIF1A Q16665 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HNF4A P41235 2/20 0.45
MCL1 Q07820 2/20 0.45
DHFR P00374 1/20 0.45
BACE1 P56817 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27450141 0.89 PARP1 (0.64) ALDH1A1DHODHPARP1BACE1
SCHEMBL902623 0.84 ALDH1A1 (0.66) ALDH1A1DHODHTP53CYP1A2HSD17B10
SCHEMBL7568063 0.81 ALDH1A1 (0.49) ALDH1A1DHODH
SCHEMBL7566766 0.81 MEN1 (0.60) ALDH1A1PARP1HSD17B10
SCHEMBL7569493 0.81 ALDH1A1 (0.49) ALDH1A1DHODHHSD17B10MCL1
SCHEMBL7575249 0.81 ALDH1A1 (0.49) ALDH1A1DHODHTP53CYP1A2HIF1A
SCHEMBL7024435 0.78 AOX1 (0.74) ALDH1A1HSD17B10
SCHEMBL7566734 0.77 KDM4E (0.51) ALDH1A1PARP1HSD17B10
SCHEMBL7030651 0.77 MEN1 (0.53) ALDH1A1PARP1TP53CYP1A2
SCHEMBL7572783 0.77 ALDH1A1 (0.45) ALDH1A1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1116285-C Bis(acridinecarboxamide) and Bis(phenazinecarboxamide) as antitumour agents XENOVA LTD (GB) 2003-07-30 CN disclosed
EP-0934278-B1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LTD (GB) 2002-09-04 EP disclosed
US-6114332-A BACTERICIDES XENOVA LIMITED (GB) 2000-09-05 US disclosed
CN-1240430-A Bis(acridinecarboxamide) and Bis(phenazinecarboxamide) as antitumour agents XENOVA LTD (GB) 2000-01-05 CN disclosed
EP-0934278-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1999-08-11 EP disclosed
WO-1998017650-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1998-04-30 WO disclosed