SCHEMBL7575249

SCHEMBL7575249

O=C(O)c1cccc2cc3cc(Cl)ccc3nc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
CYP2C9 P11712 2/20 0.44
PTGES O14684 1/20 0.44
ALOX5 P09917 1/20 0.44
HPGD P15428 1/20 0.44
CASP7 P55210 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.44
AOX1 Q06278 1/20 0.43
GRIK1 P39086 1/20 0.43
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
CASP1 P29466 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
DHODH Q02127 3/20 0.41
RXFP1 Q9HBX9 1/20 0.41
HSP90AA1 P07900 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7567042 0.88 ALDH1A1 (0.49) ALDH1A1CYP2C9PTGESALOX5HPGD
SCHEMBL27544144 0.87 PARP1 (0.51) ALDH1A1AOX1KDM4E
SCHEMBL902623 0.82 ALDH1A1 (0.66) ALDH1A1CYP2C9HPGDHSD17B10TP53
SCHEMBL7569493 0.82 ALDH1A1 (0.49) ALDH1A1HPGDHSD17B10AOX1DHODH
SCHEMBL7568063 0.82 ALDH1A1 (0.49) ALDH1A1AOX1TSHRDHODHRXFP1
SCHEMBL7566766 0.82 MEN1 (0.60) ALDH1A1HSD17B10AOX1CA1CA2
SCHEMBL7569359 0.81 ALDH1A1 (0.51) ALDH1A1HIF1AHSD17B10TP53DHODH
SCHEMBL8415114 0.79 HDAC1 (0.64) ALOX5AOX1KDM4EKMT2A
SCHEMBL7572068 0.79 ALDH1A1 (0.71) ALDH1A1CYP2C9PTGESALOX5HPGD
SCHEMBL7565784 0.79 ALDH1A1 (0.71) ALDH1A1CYP2C9PTGESALOX5HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1116285-C Bis(acridinecarboxamide) and Bis(phenazinecarboxamide) as antitumour agents XENOVA LTD (GB) 2003-07-30 CN disclosed
EP-0934278-B1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LTD (GB) 2002-09-04 EP disclosed
US-6114332-A BACTERICIDES XENOVA LIMITED (GB) 2000-09-05 US disclosed
CN-1240430-A Bis(acridinecarboxamide) and Bis(phenazinecarboxamide) as antitumour agents XENOVA LTD (GB) 2000-01-05 CN disclosed
EP-0934278-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1999-08-11 EP disclosed
WO-1998017650-A1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LIMITED (GB) 1998-04-30 WO disclosed