SCHEMBL7569982

SCHEMBL7569982

CC(C)C[C@H](NC(=O)c1ccc(-c2csc(C3=CN(C)CC=C3)n2)cc1)C(=O)N(C)C#N

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSB P07858 8/20 0.44
CTSK P43235 12/20 0.42
CTSS P25774 8/20 0.42
CTSL P07711 7/20 0.42
NPC1 O15118 2/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CAPN1 P07384 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
AGTR1 P30556 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7539652 0.89 CTSB (0.41) CTSBCTSKCTSSCTSLNPC1
SCHEMBL7486617 0.88 CTSB (0.45) CTSBCTSKCTSSCTSLNPC1
SCHEMBL7515230 0.82 CTSB (0.52) CTSBCTSKCTSSCTSLNPC1
SCHEMBL7565024 0.81 CTSB (0.41) CTSBCTSKCTSSCTSLNPC1
SCHEMBL7539033 0.80 CTSB (0.44) CTSBCTSKCTSSCTSLCAPN1
SCHEMBL6185994 0.80 CTSB (0.54) CTSBCTSKCTSSCTSLNPC1
SCHEMBL7450076 0.80 CTSB (0.54) CTSBCTSKCTSSCTSLNPC1
SCHEMBL7450318 0.80 CTSB (0.54) CTSBCTSKCTSSCTSLCAPN1
SCHEMBL7494273 0.79 CTSB (0.50) CTSBCTSKCTSSCTSLNPC1
SCHEMBL7540238 0.79 CTSK (0.58) CTSBCTSKCTSSCTSLNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO claimed