SCHEMBL7570657

SCHEMBL7570657

CO/N=C(\C)c1cc(F)ccc1F.CO/N=C(\C)c1ccc(Cl)c(F)c1.CO/N=C(\C)c1ccc(F)cc1Br

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.39
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
SLC6A4 P31645 1/20 0.34
MDM2 Q00987 5/20 0.33
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.32
PTBP1 P26599 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7782578 0.92 RAB9A (0.45) RAB9AMEN1POLBKMT2ACA12
SCHEMBL7868304 0.91 CA12 (0.34) RAB9AMEN1POLBKMT2ACA12
SCHEMBL7844833 0.89 RAB9A (0.42) RAB9AMEN1POLBKMT2ACA12
SCHEMBL7777665 0.81 SMN1; SMN2 (0.38) RAB9AMEN1POLBKMT2ACA12
SCHEMBL6811367 0.80 SLC6A4 (0.45) RAB9AMEN1POLBKMT2ACA12
SCHEMBL6815992 0.80 TRPA1 (0.39) RAB9AMEN1POLBKMT2AMAPT
SCHEMBL6815999 0.80 TRPA1 (0.39) RAB9AMEN1POLBKMT2AMAPT
SCHEMBL6811369 0.80 SLC6A4 (0.45) RAB9AMEN1POLBKMT2ACA12
SCHEMBL6819076 0.78 CES2 (0.47) RAB9AMEN1POLBKMT2ACA9
SCHEMBL6819080 0.78 CES2 (0.47) RAB9AMEN1POLBKMT2ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144399-A3 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP Wyeth (US) 2002-09-11 EP disclosed
EP-1144399-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-17 EP disclosed
WO-2000034261-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed