SCHEMBL7570905

SCHEMBL7570905

Cc1cc(C2=NC(Cc3ccc(-c4ccccc4)cc3)C(=O)N=C2O)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 1/20 0.35
CNR2 P34972 3/20 0.33
HDAC3 O15379 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
SUCNR1 Q9BXA5 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
KDM4A O75164 1/20 0.32
KDM5A P29375 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
CXCR2 P25025 2/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
MMP1 P03956 1/20 0.32
MMP7 P09237 1/20 0.32
MMP9 P14780 1/20 0.32
MMP8 P22894 1/20 0.32
MMP13 P45452 1/20 0.32
PTPN5 P54829 1/20 0.32
CES2 O00748 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7576399 0.96 CNR2 (0.35) CNR2HDAC3HDAC6PDE3BPDE3A
SCHEMBL7571399 0.90 PTPN5 (0.38) CYP26A1HDAC3HDAC6ESR2PTPN5
SCHEMBL7570886 0.85 PSD (0.37) HDAC3HDAC6CXCR2PTPN5
SCHEMBL7571248 0.85 HDAC3 (0.41) CYP26A1HDAC3HDAC6
SCHEMBL7572718 0.84 CES2 (0.43) HDAC3HDAC6CES2
SCHEMBL7572646 0.82 BDKRB2 (0.41) CYP26A1HDAC3HDAC6CES2
SCHEMBL7575515 0.82 ESR1 (0.37) CYP26A1HDAC3HDAC6ESR1ESR2
SCHEMBL7572458 0.80 BDKRB2 (0.42) HDAC3HDAC6CES2
SCHEMBL7572631 0.79 CES2 (0.42) CYP26A1HDAC3HDAC6MMP1MMP9
SCHEMBL7576544 0.79 CES2 (0.44) HDAC3HDAC6CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002085369-A1 INHIBITORS OF ANTHRAX LETHAL FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS, INC. (US) 2002-10-31 WO disclosed