SCHEMBL7571248

SCHEMBL7571248

O=C1N=C(O)C(c2ccc(-c3ccccc3)cc2)=NC1Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
BDKRB2 P30411 5/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
CYP26A1 O43174 1/20 0.37
ABCC4 O15439 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
PTGS1 P23219 1/20 0.37
HTT P42858 1/20 0.37
FFAR1 O14842 1/20 0.35
SLC13A5 Q86YT5 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
GPR84 Q9NQS5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572646 0.97 BDKRB2 (0.41) HDAC3HDAC6BDKRB2HDAC1HDAC8
SCHEMBL7572458 0.94 BDKRB2 (0.42) HDAC3HDAC6BDKRB2HDAC1HDAC8
SCHEMBL7572631 0.94 CES2 (0.42) HDAC3HDAC6BDKRB2HDAC1HDAC8
SCHEMBL7572718 0.94 CES2 (0.43) HDAC3HDAC6BDKRB2HDAC1HDAC8
SCHEMBL7570328 0.90 CES2 (0.45) HDAC3HDAC6LMNAHTTFFAR1
SCHEMBL7571381 0.90 HDAC3 (0.42) HDAC3HDAC6BDKRB2HDAC1HDAC8
SCHEMBL7575515 0.89 ESR1 (0.37) HDAC3HDAC6HDAC8CYP26A1LMNA
SCHEMBL7576544 0.88 CES2 (0.44) HDAC3HDAC6BDKRB2HDAC1HDAC8
SCHEMBL7571711 0.88 CES2 (0.38) HDAC3HDAC6BDKRB2HDAC1HDAC8
SCHEMBL7571208 0.88 NPC1 (0.44) HDAC3HDAC6BDKRB2HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002085369-A1 INHIBITORS OF ANTHRAX LETHAL FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS, INC. (US) 2002-10-31 WO disclosed