SCHEMBL7571479

SCHEMBL7571479

Cc1c[nH]c(C(=O)c2ccc(N)cc2Cl)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.44
TYK2 P29597 1/20 0.44
ALDH1A1 P00352 3/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 2/20 0.39
CHRM2 P08172 1/20 0.38
CHRM3 P20309 1/20 0.38
MAOA P21397 1/20 0.38
HTR2C P28335 1/20 0.38
CHRNA4 P43681 1/20 0.38
HTR3A P46098 1/20 0.38
KCNH2 Q12809 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
CYP3A4 P08684 2/20 0.38
HTT P42858 1/20 0.37
MAPK13 O15264 2/20 0.36
MAPK12 P53778 2/20 0.36
MAPK11 Q15759 2/20 0.36
MAPK14 Q16539 2/20 0.36
NR1H4 Q96RI1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7565415 0.79 MAPK14 (0.65) MAPK13MAPK12MAPK11MAPK14MAPT
SCHEMBL7571478 0.75 MAPK14 (0.67) MAPK13MAPK12MAPK11MAPK14KMT2A
SCHEMBL7090488 0.75 JAK2 (0.53) JAK2TYK2ALDH1A1KDM4ECHRM2
SCHEMBL8307733 0.74 KMT2A (0.64) JAK2TYK2ALDH1A1CHRM2CHRM3
SCHEMBL9038897 0.74 GAA (0.46) ALDH1A1KDM4EMAPK13MAPK12MAPK11
SCHEMBL5151745 0.73 NPC1 (0.32) NPC1RAB9A
Bromide SCHEMBL7429002 0.71 NPC1 (0.32) NPC1RAB9A
SCHEMBL7563806 0.71 MAPK13 (0.68) ALDH1A1LMNAHTTMAPK13MAPK12
SCHEMBL29088628 0.70 MAPT (0.51) JAK2TYK2ALDH1A1LMNACYP3A4
SCHEMBL7035012 0.70 CYP3A4 (0.48) JAK2TYK2ALDH1A1LMNACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002083622-A2 NOVEL AMINOPHENYL KETONE DERIVATIVES LEO PHARMA A/S (DK) 2002-10-24 WO disclosed