SCHEMBL7571567

SCHEMBL7571567

O=S(=O)(Nc1ccc(Br)c(Br)c1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 1/20 0.63
NR3C1 P04150 1/20 0.61
PGR P06401 1/20 0.61
AR P10275 1/20 0.61
ESR2 Q92731 1/20 0.61
TSHR P16473 1/20 0.59
HDAC1 Q13547 1/20 0.58
HDAC8 Q9BY41 1/20 0.58
CA2 P00918 2/20 0.56
CA1 P00915 1/20 0.56
MMP1 P03956 1/20 0.56
MMP2 P08253 1/20 0.56
MMP9 P14780 1/20 0.56
MMP8 P22894 1/20 0.56
MMP13 P45452 1/20 0.56
FFAR1 O14842 1/20 0.56
CDK1 P06493 1/20 0.56
CCNB1 P14635 1/20 0.56
CCNA2 P20248 1/20 0.56
CDK2 P24941 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19065106 0.84 TSHR (0.64) HSD17B2NR3C1PGRARESR2
SCHEMBL7591899 0.84 KMT2A (0.61) HSD17B2NR3C1PGRARESR2
SCHEMBL22441723 0.82 CDK1 (0.64) HSD17B2NR3C1PGRARESR2
SCHEMBL7572806 0.81 NR3C1 (0.69) HSD17B2NR3C1PGRARESR2
SCHEMBL3762909 0.81 PGR (0.77) HSD17B2NR3C1PGRARESR2
SCHEMBL7573925 0.81 HSD17B2 (0.79) HSD17B2NR3C1PGRARESR2
SCHEMBL7825221 0.81 TSHR (0.62) HSD17B2NR3C1PGRARESR2
SCHEMBL7572556 0.80 PGR (0.67) HSD17B2NR3C1PGRARESR2
SCHEMBL97543 0.80 NR3C1 (0.67) HSD17B2NR3C1PGRARESR2
SCHEMBL7571512 0.78 KMT2A (0.60) HSD17B2PGRHDAC1HDAC8KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1239852-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS Arrow Therapeutics Limited (GB) 2002-09-18 EP disclosed
WO-2001028537-A2 BISSULFONAMIDE DERIVATIVES AS ENZYME INHIBITORS ARROW THERAPEUTICS LIMITED (GB) 2001-04-26 WO disclosed