SCHEMBL7579606

SCHEMBL7579606

COc1ccc(C#CCN=Cc2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.45
G6PC1 P35575 1/20 0.43
APP P05067 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
FAAH O00519 1/20 0.40
POLB P06746 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
KCNH2 Q12809 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP13 P45452 1/20 0.39
THRB P10828 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7579599 1.00 TRPA1 (0.45) TRPA1G6PC1APPNPC1RAB9A
SCHEMBL7572532 0.86 MAOB (0.39) APPNPC1RAB9APOLBALDH1A1
SCHEMBL7572529 0.86 MAOB (0.39) APPNPC1RAB9APOLBALDH1A1
SCHEMBL7571246 0.84 CYP1A2 (0.45) G6PC1APPPOLBALDH1A1MAPT
SCHEMBL7571250 0.84 CYP1A2 (0.45) G6PC1APPPOLBALDH1A1MAPT
SCHEMBL7573177 0.84 RELA (0.51) NPC1RAB9AMAPTKCNH2GAA
SCHEMBL7573181 0.84 RELA (0.51) NPC1RAB9AMAPTKCNH2GAA
SCHEMBL7581846 0.83 MAPT (0.47) NPC1RAB9APOLBALDH1A1MAPT
SCHEMBL7581838 0.83 MAPT (0.47) NPC1RAB9APOLBALDH1A1MAPT
SCHEMBL7574544 0.81 NFE2L2 (0.47) APPPOLBALDH1A1MAPTKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed