SCHEMBL7573441

SCHEMBL7573441

C#C/C(N)=C\c1ccc(Cl)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.51
GABRG2 P18507 2/20 0.51
GABRB3 P28472 2/20 0.51
MAPT P10636 4/20 0.47
GRIN2D O15399 2/20 0.47
GRIN3B O60391 2/20 0.47
GRIN1 Q05586 2/20 0.47
GRIN2A Q12879 2/20 0.47
GRIN2B Q13224 2/20 0.47
GRIN2C Q14957 2/20 0.47
GRIN3A Q8TCU5 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7571231 0.79 TRPA1 (0.53) MAPTGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8262436 0.79 MAPT (0.59) GABRA1GABRG2GABRB3MAPTGRIN2D
SCHEMBL8272588 0.76 GABRA1 (0.61) GABRA1GABRG2GABRB3MAPTGRIN2D
SCHEMBL7575165 0.73 GRIN2D (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL7575017 0.71 GRIN1 (0.47) MAPTGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6340710 0.71 GABRA1 (0.55) GABRA1GABRG2GABRB3MAPTGRIN2D
SCHEMBL3226151 0.71 TDP1 (0.54) GABRA1GABRG2GABRB3MAPTGRIN2D
SCHEMBL272063 0.70 GABRA1 (0.69) GABRA1GABRG2GABRB3MAPTGRIN2D
SCHEMBL4849644 0.69 TDP1 (0.57) GABRA1GABRG2GABRB3MAPTGRIN2D
SCHEMBL29028260 0.68 GABRA1 (0.61) GABRA1GABRG2GABRB3MAPTGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810199-B1 Method for producing propargylamine compounds SUMITOMO CHEMICAL CO (JP) 2002-09-25 EP disclosed
US-5756769-A Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1998-05-26 US disclosed
EP-0810199-A1 Method for producing propargylamine compounds SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-12-03 EP disclosed