SCHEMBL7574640

SCHEMBL7574640

CCC(=NOC)c1ccc(F)cc1.CON=CCc1cccc(Br)c1.CON=CCc1cccc(Cl)c1.CON=CCc1ccccc1Cl

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
GRIN2B Q13224 1/20 0.33
DRD4 P21917 8/20 0.32
DRD2 P14416 5/20 0.32
GSK3B P49841 1/20 0.31
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864156 0.86 DRD4 (0.39) LMNAPOLBMEN1ALDH1A1KMT2A
SCHEMBL7778596 0.75 GRIN2B (0.38) LMNAPOLBCYP1A2CYP2C19MEN1
SCHEMBL7861405 0.75 PPARG (0.39) LMNAPOLBCYP1A2CYP2D6CYP2C9
SCHEMBL6811236 0.66 TRPA1 (0.49) LMNAMEN1KMT2ADRD4DRD2
SCHEMBL27548769 0.65 GSK3B (0.49) CYP1A2GSK3BGAA
SCHEMBL28113822 0.64 ALDH1A1 (0.57) LMNACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7569694 0.63 MAOB (0.38) LMNAPOLBMEN1ALDH1A1KMT2A
SCHEMBL7844834 0.63 GCGR (0.33) LMNAALDH1A1DRD4DRD2MAPT
SCHEMBL27469352 0.62 DRD4 (0.49) CYP1A2CYP2D6CYP2C9CYP2C19MEN1
SCHEMBL7575131 0.62 AKR1B1 (0.36) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144399-A3 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP Wyeth (US) 2002-09-11 EP disclosed
EP-1144399-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-17 EP disclosed
WO-2000034261-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed