SCHEMBL7575469

SCHEMBL7575469

CCCCC(=O)Nc1ccc(C(=O)O)cc1NCc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 2/20 0.44
LTB4R2 Q9NPC1 2/20 0.43
HTT P42858 1/20 0.41
SOAT1 P35610 2/20 0.40
AGTR1 P30556 4/20 0.40
AGTR2 P50052 2/20 0.40
LTB4R Q15722 1/20 0.39
GSK3A P49840 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7570389 0.86 HTT (0.40) LTB4R2HTTSOAT1LTB4RGSK3A
SCHEMBL7570660 0.85 PTGER1 (0.41) BDKRB1SOAT1LTB4R
SCHEMBL7570385 0.83 SOAT1 (0.40) BDKRB1LTB4R2HTTSOAT1GSK3A
SCHEMBL7575457 0.83 SOAT1 (0.40) BDKRB1LTB4R2HTTSOAT1AGTR1
SCHEMBL8081241 0.80 BDKRB1 (0.44) BDKRB1LTB4R2SOAT1AGTR1AGTR2
SCHEMBL4609709 0.80 LTB4R2 (0.60) BDKRB1LTB4R2HTT
SCHEMBL7567767 0.80 HTT (0.51) HTTLTB4R
SCHEMBL9709600 0.77 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL7570411 0.75 POLB (0.47) BDKRB1HTTLTB4R
SCHEMBL9263754 0.75 AGTR1 (0.44) BDKRB1AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685470-B1 Benzene derivatives and pharmaceutical composition KUREHA CHEMICAL IND CO LTD (JP) 2002-09-11 EP disclosed
EP-0685470-A2 Benzene derivatives and pharmaceutical composition Kureha Chemical Industry Co., Ltd. (JP) 1995-12-06 EP disclosed