SCHEMBL7575928

SCHEMBL7575928

CON=C(C)c1cccc(C(F)(F)F)c1.CON=CCc1ccc(F)cc1F.CON=CCc1ccccc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 2/20 0.37
NPSR1 Q6W5P4 2/20 0.36
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
DDR1 Q08345 4/20 0.34
GAA P10253 1/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
HIF1A Q16665 1/20 0.33
POLB P06746 1/20 0.32
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7575921 0.78 KMT2A (0.42) NPSR1KMT2AMEN1GAAKDM4E
SCHEMBL7846221 0.77 KMT2A (0.43) NPSR1KMT2AMEN1GAAPOLB
SCHEMBL7866288 0.75 EPHX2 (0.38) KMT2AGAAMAPTPOLB
SCHEMBL7861383 0.74 HIF1A (0.39) KMT2AMEN1KDM4EMAPTHIF1A
SCHEMBL6819739 0.74 KMT2A (0.57) NPSR1KMT2AMEN1GAAMAPT
SCHEMBL29778306 0.74 KMT2A (0.57) NPSR1KMT2AMEN1GAAMAPT
SCHEMBL6819302 0.74 KMT2A (0.57) NPSR1KMT2AMEN1GAAMAPT
SCHEMBL7569653 0.74 IDO1 (0.50) KMT2AMEN1KDM4EPOLB
SCHEMBL7868617 0.73 S1PR1 (0.34) KMT2AMEN1S1PR1S1PR3
SCHEMBL7868713 0.72 MAOB (0.46) NPSR1KMT2AMEN1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144399-A3 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP Wyeth (US) 2002-09-11 EP disclosed
EP-1144399-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-17 EP disclosed
WO-2000034261-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A SUBSTITUTED PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed