SCHEMBL7581886

SCHEMBL7581886

C=C1[C@@H](c2ccc(C(F)(F)F)cc2)[C@@](C)(c2cccc(C(F)(F)F)c2)NC(=N)N1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.34
AR P10275 2/20 0.33
OPRL1 P41146 2/20 0.33
HTT P42858 2/20 0.32
CCR2 P41597 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PGR P06401 2/20 0.32
LMNA P02545 2/20 0.31
HCAR3 P49019 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
ESR1 P03372 1/20 0.31
NR3C1 P04150 1/20 0.31
NR3C2 P08235 1/20 0.31
ESR2 Q92731 1/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
SLC6A2 P23975 1/20 0.31
TEAD1 P28347 1/20 0.31
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7582110 0.95 KDM1A (0.33) KDM1AARHTTCCR2TEAD1
SCHEMBL7588738 0.92 PAX8 (0.31) MEN1KMT2APGR
SCHEMBL7588393 0.92 P2RX7 (0.34) MEN1KMT2APGRSLC6A4
SCHEMBL7583661 0.91 PGR (0.31) HTTMEN1KMT2APGRSLC6A4
SCHEMBL7583857 0.89 HTT (0.34) HTTOPRK1
SCHEMBL7582989 0.89
SCHEMBL7588502 0.89 MEN1 (0.31) MEN1KMT2AESR1
SCHEMBL7583245 0.88
SCHEMBL7584231 0.88 ELANE (0.33) HTT
SCHEMBL7579123 0.87 NR1H2 (0.37) MEN1KMT2AESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed