SCHEMBL7583857

SCHEMBL7583857

C=C1[C@@H](c2ccc(C(F)(F)F)cc2)[C@@](C)(c2cccc(CC)c2)NC(=N)N1C

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.34
OPRK1 P41145 1/20 0.30
MAPT P10636 1/20 0.30
ATM Q13315 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7588871 0.93
SCHEMBL7581886 0.89 KDM1A (0.34) HTTOPRK1
SCHEMBL7554785 0.88 HTT (0.36) HTTSMN1; SMN2
SCHEMBL13055115 0.88 HTT (0.36) HTTSMN1; SMN2
SCHEMBL7588738 0.87 PAX8 (0.31)
SCHEMBL7588393 0.87 P2RX7 (0.34)
SCHEMBL7583661 0.86 PGR (0.31) HTTMAPTATM
SCHEMBL7588502 0.84 MEN1 (0.31)
SCHEMBL7582989 0.84
SCHEMBL7582110 0.84 KDM1A (0.33) HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed