SCHEMBL7582205

SCHEMBL7582205

CCC(F)c1cc(N2CCN(CCO)CC2)cc(-c2ccccc2C)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.38
DRD3 P35462 1/20 0.38
MAPT P10636 3/20 0.37
HTR1A P08908 3/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HRH4 Q9H3N8 1/20 0.36
METAP1 P53582 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
LMNA P02545 2/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HTR2A P28223 1/20 0.34
HTR7 P34969 1/20 0.34
ADRA1A P35348 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7585740 0.92 DRD2 (0.44) DRD2DRD3HTR1ALMNASIGMAR1
SCHEMBL7583679 0.91 DRD2 (0.44) DRD2DRD3MAPTHTR1ANPSR1
SCHEMBL7585162 0.89 CHRNA7 (0.42) MAPTHTR1ALMNAKDM4EALDH1A1
SCHEMBL7587432 0.89 MAPT (0.39) DRD2DRD3MAPTHTR1ANPSR1
SCHEMBL7591499 0.88 TACR1 (0.39) DRD2DRD3HTR1ALMNAMAPK1
SCHEMBL7584119 0.88 TACR1 (0.39) DRD2DRD3HTR1ALMNAMAPK1
SCHEMBL7585760 0.88 TACR1 (0.39) DRD2DRD3HTR1ALMNAMAPK1
SCHEMBL7955784 0.87 MAPT (0.38) DRD2DRD3MAPTNPSR1HRH4
SCHEMBL7584122 0.87 MAPT (0.38) DRD2DRD3MAPTNPSR1HRH4
SCHEMBL7589752 0.86 DRD2 (0.36) DRD2DRD3MAPTHTR1ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0675118-B1 Biphenylderivatives, process for their preparation and their use as medicaments EISAI CO LTD (JP) 2002-10-09 EP claimed
EP-0675118-A2 Biphenylderivatives, process for their preparation and their use as medicaments Eisai Co., Ltd. (JP) 1995-10-04 EP claimed
EP-0675118-B1 Biphenylderivatives, process for their preparation and their use as medicaments EISAI CO LTD (JP) 2002-10-09 EP disclosed
US-6281214-B1 USEFUL FOR TREATING AND AMELIORATING MENTAL DISORDERS EISAI CO., LTD (JP) 2001-08-28 US disclosed
EP-0675118-A2 Biphenylderivatives, process for their preparation and their use as medicaments Eisai Co., Ltd. (JP) 1995-10-04 EP disclosed