SCHEMBL7582359

SCHEMBL7582359

C=C1[C@@H](c2ccc(N(C)S(C)(=O)=O)cc2)[C@@](C)(c2cccc(C#N)c2)NC(=N)N1C

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.36
NR1H3 Q13133 1/20 0.32
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13054511 0.90 PGR (0.37) PGRNR1H3BACE1
SCHEMBL7572682 0.90 PGR (0.37) PGRNR1H3BACE1
SCHEMBL7582435 0.86 BACE1 (0.34) PGRBACE1
SCHEMBL7584784 0.84 RORC (0.33) BACE1
SCHEMBL7589711 0.83 ATR (0.32) BACE1
SCHEMBL7584770 0.83 BACE1 (0.32) BACE1
SCHEMBL7584411 0.82 KMT2A (0.32) BACE1
SCHEMBL7584371 0.81 BACE1 (0.31) BACE1
SCHEMBL7584231 0.81 ELANE (0.33) BACE1
SCHEMBL7581190 0.80 BACE1 (0.31) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8183252-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-22 US disclosed