SCHEMBL7583097

SCHEMBL7583097

CCOc1ccc(C(=O)c2c(Cl)cc(Cl)cc2Cl)cc1Cc1ccc(=O)[nH]n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
MAPT P10636 2/20 0.40
CYP3A4 P08684 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
CYP1A2 P05177 3/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CYP2C19 P33261 2/20 0.39
TP53 P04637 1/20 0.39
CYP2D6 P10635 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
USP2 O75604 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
F10 P00742 1/20 0.37
LMNA P02545 1/20 0.36
ADRB2 P07550 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7590797 0.92 L3MBTL1 (0.40) ALDH1A1MAPTCYP3A4SMN1; SMN2CYP1A2
SCHEMBL7585660 0.90 ADRB2 (0.44) ALDH1A1MAPK1MAPTCYP3A4SMN1; SMN2
SCHEMBL7584283 0.87 GAA (0.40) ALDH1A1CYP3A4CYP1A2NPC1RAB9A
SCHEMBL7583126 0.87 ADRB2 (0.39) ALDH1A1MAPK1MAPTCYP3A4L3MBTL1
SCHEMBL7589686 0.85 CYP3A4 (0.44) CYP3A4LMNA
SCHEMBL7583539 0.84 CYP3A4 (0.42) MAPTCYP3A4NPC1RAB9AHDAC1
SCHEMBL7582260 0.83 CYP3A4 (0.42) CYP3A4SMN1; SMN2LMNAMRGPRX4
SCHEMBL7583085 0.83 CYP3A4 (0.45) ALDH1A1MAPTCYP3A4SMN1; SMN2CYP1A2
SCHEMBL7584819 0.82 ADRB2 (0.39) ALDH1A1MAPK1MAPTCYP3A4SMN1; SMN2
SCHEMBL7587071 0.82 CYP3A4 (0.42) CYP3A4LMNAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810218-B1 6-Benzyl-2H-pyridazin-3-one derivatives,their preparation and their use as inhibitors of prostaglandin G/H synthase I and II (COX I and COX II) HOFFMANN LA ROCHE (CH) 2002-12-04 EP disclosed
EP-0810218-A1 6-Benzyl-2H-pyridazin-3-one derivatives,their preparation and their use as inhibitors of prostaglandin G/H synthase I and II (COX I and COX II) F. HOFFMANN-LA ROCHE AG (CH) 1997-12-03 EP disclosed