SCHEMBL7583389

SCHEMBL7583389

CCCc1cc(N2CCN(CC)CC2)cc(-c2ccccc2C)c1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.43
CHRNA7 P36544 1/20 0.43
KMT2A Q03164 2/20 0.40
MAPT P10636 3/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 1/20 0.40
ALOX15 P16050 1/20 0.40
GAA P10253 2/20 0.40
RAD52 P43351 2/20 0.40
DRD2 P14416 4/20 0.38
POLB P06746 1/20 0.37
DRD4 P21917 2/20 0.36
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36
DRD3 P35462 1/20 0.36
HTR1A P08908 1/20 0.36
KHK P50053 1/20 0.35
KDM4E B2RXH2 1/20 0.35
GFER P55789 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7583334 0.89 HTR7 (0.46) HTR7CHRNA7KMT2AMAPTLMNA
SCHEMBL7581209 0.88 HTR7 (0.44) HTR7CHRNA7KMT2AMAPTLMNA
SCHEMBL7583969 0.86 CHRNA7 (0.48) HTR7CHRNA7KMT2AMAPTLMNA
SCHEMBL7582076 0.81 DRD2 (0.47) HTR7CHRNA7KMT2AMAPTLMNA
SCHEMBL7584847 0.80 SMN1; SMN2 (0.40) HTR7CHRNA7MAPTLMNAALOX15
SCHEMBL7593291 0.80 LMNA (0.44) CHRNA7KMT2AMAPTLMNAMEN1
SCHEMBL7586646 0.79 KDM4E (0.40) HTR7CHRNA7MAPTLMNAALOX15
SCHEMBL7584437 0.78 CHRNA7 (0.47) HTR7CHRNA7KMT2AMAPTLMNA
SCHEMBL7586374 0.77 CHRNA7 (0.46) HTR7CHRNA7KMT2AMAPTLMNA
SCHEMBL7582907 0.77 KDM4E (0.42) HTR7CHRNA7MAPTLMNAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0675118-B1 Biphenylderivatives, process for their preparation and their use as medicaments EISAI CO LTD (JP) 2002-10-09 EP claimed
EP-0675118-A2 Biphenylderivatives, process for their preparation and their use as medicaments Eisai Co., Ltd. (JP) 1995-10-04 EP claimed
EP-0675118-B1 Biphenylderivatives, process for their preparation and their use as medicaments EISAI CO LTD (JP) 2002-10-09 EP disclosed
US-6281214-B1 USEFUL FOR TREATING AND AMELIORATING MENTAL DISORDERS EISAI CO., LTD (JP) 2001-08-28 US disclosed
EP-0675118-A2 Biphenylderivatives, process for their preparation and their use as medicaments Eisai Co., Ltd. (JP) 1995-10-04 EP disclosed