SCHEMBL7584062

SCHEMBL7584062

CCN1CCN(c2cc(-c3ccccc3C)c(Cl)c(S(=O)(=O)N(C)C)c2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.43
MAPT P10636 3/20 0.43
ALDH1A1 P00352 4/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
MAPK1 P28482 1/20 0.41
CHRNA7 P36544 1/20 0.40
KDM2B Q8NHM5 3/20 0.40
MITF O75030 1/20 0.39
KDM4E B2RXH2 1/20 0.38
DRD3 P35462 3/20 0.38
HRH3 Q9Y5N1 2/20 0.38
APAF1 O14727 1/20 0.38
RAD52 P43351 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CNR1 P21554 2/20 0.37
CNR2 P34972 2/20 0.37
HTR6 P50406 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7585774 0.88 CHRNA7 (0.43) GAAKMT2ACHRNA7KDM2BMITF
SCHEMBL7583617 0.85 CHRNA7 (0.40) GAAKMT2ACHRNA7KDM2BMITF
SCHEMBL7583056 0.84 SMN1; SMN2 (0.41) GAAMAPTMEN1KMT2APOLB
SCHEMBL7586735 0.82 MITF (0.41) GAAPOLBCHRNA7KDM2BMITF
SCHEMBL7581561 0.82 APAF1 (0.44) MAPTALDH1A1MEN1KMT2ACHRNA7
SCHEMBL8629280 0.79 MITF (0.41) GAACHRNA7KDM2BMITFKDM4E
SCHEMBL7583496 0.78 GAA (0.52) GAAMAPTMEN1KMT2ACHRNA7
SCHEMBL7583743 0.77 CHRNA7 (0.43) GAAMAPTKMT2APOLBCHRNA7
SCHEMBL7583735 0.77 CHRNA7 (0.44) GAAMAPTKMT2ACHRNA7KDM4E
SCHEMBL8627347 0.76 MITF (0.39) GAACHRNA7MITFDRD3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0675118-B1 Biphenylderivatives, process for their preparation and their use as medicaments EISAI CO LTD (JP) 2002-10-09 EP claimed
EP-0675118-A2 Biphenylderivatives, process for their preparation and their use as medicaments Eisai Co., Ltd. (JP) 1995-10-04 EP claimed
EP-0675118-B1 Biphenylderivatives, process for their preparation and their use as medicaments EISAI CO LTD (JP) 2002-10-09 EP disclosed
US-6281214-B1 USEFUL FOR TREATING AND AMELIORATING MENTAL DISORDERS EISAI CO., LTD (JP) 2001-08-28 US disclosed
US-5849912-A Biphenyl derivatives EISAI CO., LTD. (JP) 1998-12-15 US disclosed
EP-0675118-A2 Biphenylderivatives, process for their preparation and their use as medicaments Eisai Co., Ltd. (JP) 1995-10-04 EP disclosed