SCHEMBL7584586

SCHEMBL7584586

CC(C)Oc1ccc(C(C)(C)C#N)cc1C=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 1/20 0.36
MAPT P10636 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ERN1 O75460 1/20 0.33
DHODH Q02127 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A3 P47895 1/20 0.33
XDH P47989 1/20 0.32
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
VEGFA P15692 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALK Q9UM73 1/20 0.30
SYK P43405 1/20 0.30
CTSA P10619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7587116 0.84 ALDH1A1 (0.44) ERN1DHODHL3MBTL1KDM4EALDH1A1
SCHEMBL8327036 0.77 CYP1A2 (0.40) MAPTCYP1A2CYP2C9CYP2C19ERN1
SCHEMBL13755069 0.77 MAPT (0.38) MAPTCYP1A2CYP2C9CYP2C19ERN1
SCHEMBL307932 0.73 ALDH1A1 (0.39) SCN10ACYP1A2CYP2C9CYP2C19ERN1
SCHEMBL28340475 0.73 MAPT (0.39) MAPTCYP1A2CYP2C9CYP2C19L3MBTL1
SCHEMBL7591958 0.73 ALDH1A1 (0.46) ERN1L3MBTL1KDM4EALDH1A1TSHR
SCHEMBL6098469 0.72 ERN1 (0.45) SCN10AMAPTERN1XDHKDM4E
SCHEMBL6930848 0.72 ALDH1A3 (0.53) MAPTCYP1A2CYP2C9CYP2C19ERN1
SCHEMBL5651250 0.71 TYR (0.45) SCN10AMAPTERN1ALDH1A1TDP1
SCHEMBL7591252 0.70 ALDH1A1 (0.44) MAPTCYP1A2CYP2C9CYP2C19ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780375-B1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER (US) 2002-09-11 EP disclosed
US-5789423-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS; GASTROINTESTINAL AND CENTRAL NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-08-04 US disclosed
EP-0780375-A1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER INC. (US) 1997-06-25 EP disclosed