SCHEMBL7587116

SCHEMBL7587116

COc1ccc(C(C)(C)C#N)cc1C=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
TUBB1 Q9H4B7 1/20 0.40
PDE4A P27815 6/20 0.40
PDE4B Q07343 6/20 0.40
PDE4C Q08493 6/20 0.40
PDE4D Q08499 6/20 0.40
DHODH Q02127 1/20 0.39
CASP1 P29466 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LMNA P02545 2/20 0.38
PRKDC P78527 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
HPGD P15428 1/20 0.37
ERN1 O75460 2/20 0.37
TLR2 O60603 1/20 0.36
TLR1 Q15399 1/20 0.36
TLR6 Q9Y2C9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7591958 0.89 ALDH1A1 (0.46) ALDH1A1TSHRKDM4ETDP1TUBB1
SCHEMBL7591252 0.85 ALDH1A1 (0.44) ALDH1A1TSHRKDM4ETDP1TUBB1
SCHEMBL7588840 0.84 ALDH1A1 (0.44) ALDH1A1TSHRKDM4ETDP1TUBB1
SCHEMBL7584586 0.84 SCN10A (0.36) ALDH1A1TSHRKDM4ETDP1DHODH
SCHEMBL7591027 0.83 ALDH1A1 (0.47) ALDH1A1TSHRKDM4ETDP1TUBB1
SCHEMBL31738417 0.82 ALDH1A1 (0.52) ALDH1A1TSHRKDM4ETDP1TUBB1
SCHEMBL4186655 0.82 ALDH1A1 (0.52) ALDH1A1TSHRKDM4ETDP1TUBB1
SCHEMBL7591018 0.81 CASP1 (0.43) ALDH1A1TSHRKDM4ETDP1TUBB1
SCHEMBL7130351 0.81 ALDH1A1 (0.45) ALDH1A1TSHRKDM4ETDP1TUBB1
SCHEMBL601637 0.80 CASP1 (0.57) ALDH1A1TSHRKDM4EPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780375-B1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER (US) 2002-09-11 EP disclosed
US-5789423-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS; GASTROINTESTINAL AND CENTRAL NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-08-04 US disclosed
EP-0780375-A1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER INC. (US) 1997-06-25 EP disclosed