SCHEMBL7585672

SCHEMBL7585672

CN(C)CC1=C(c2cccc(O)c2)c2cc(-c3ccccc3)ccc2CC1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.46
HSD17B1 P14061 9/20 0.41
HSD17B2 P37059 9/20 0.41
TDP2 O95551 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP17A1 P05093 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
OPRD1 P41143 3/20 0.37
ESR1 P03372 1/20 0.36
SLC6A9 P48067 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8012131 0.99 OPRK1 (0.45) OPRK1HSD17B1HSD17B2TDP2CYP3A4
SCHEMBL7587708 0.90 OPRK1 (0.46) OPRK1HSD17B1HSD17B2TDP2CYP3A4
SCHEMBL7584146 0.90 PBRM1 (0.40) OPRK1HSD17B1HSD17B2TDP2CYP3A4
Hydrochloric Acid SCHEMBL8013584 0.89 OPRK1 (0.45) OPRK1HSD17B1HSD17B2TDP2CYP3A4
Hydrochloric Acid SCHEMBL8017505 0.89 PBRM1 (0.39) OPRK1HSD17B1HSD17B2TDP2CYP3A4
SCHEMBL7591741 0.87 MTNR1A (0.44) OPRK1HSD17B1HSD17B2TDP2CYP3A4
SCHEMBL7588246 0.86 OPRK1 (0.40) OPRK1HSD17B1HSD17B2OPRD1
Hydrochloric Acid SCHEMBL8010759 0.86 MTNR1A (0.43) OPRK1HSD17B1HSD17B2TDP2CYP3A4
SCHEMBL7588071 0.86 TDP2 (0.41) OPRK1HSD17B1HSD17B2TDP2CYP3A4
SCHEMBL7586089 0.85 OPRK1 (0.36) OPRK1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
CN-1197059-A Substituted amino compounds and their use as substances having analgesic effect GRUENENTHAL GMBH (DE) 1998-10-28 CN disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed