SCHEMBL7586256

SCHEMBL7586256

CCOC(=O)C(C)(N)Cc1c(CC)ccc(N)c1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
LMNA P02545 1/20 0.36
MAOA P21397 1/20 0.36
MMP8 P22894 1/20 0.35
MAPK1 P28482 2/20 0.35
ALDH1A1 P00352 3/20 0.35
HSD17B10 Q99714 2/20 0.35
ABCB11 O95342 1/20 0.35
TSHR P16473 1/20 0.35
HTR2A P28223 1/20 0.35
PMP22 Q01453 1/20 0.35
PPARA Q07869 1/20 0.35
PPIB P23284 1/20 0.35
PPIA P62937 1/20 0.35
PPID Q08752 1/20 0.35
PPIG Q13427 1/20 0.35
CNR2 P34972 2/20 0.33
PIN1 Q13526 1/20 0.33
HDAC3 O15379 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9232038 0.77 CNR2 (0.34) CYP1A2CYP3A4LMNAMAOAMMP8
SCHEMBL9233712 0.75 KDM4E (0.37) LMNAALDH1A1HSD17B10CNR2PIN1
SCHEMBL9231432 0.70 THRB (0.39) CYP3A4LMNAALDH1A1TSHRRECQL
SCHEMBL604459 0.70 MMP8 (0.61) LMNAMMP8ALDH1A1TSHRPPID
SCHEMBL10684512 0.70 MMP8 (0.61) LMNAMMP8ALDH1A1TSHRPPID
SCHEMBL1831636 0.70 MMP8 (0.61) LMNAMMP8ALDH1A1TSHRPPID
SCHEMBL571458 0.69 POLB (0.40) ALDH1A1MAPT
SCHEMBL9386398 0.69 BLM (0.63) CYP1A2CYP3A4MMP8ALDH1A1HSD17B10
SCHEMBL9386400 0.69 BLM (0.63) CYP1A2CYP3A4MMP8ALDH1A1HSD17B10
SCHEMBL7563841 0.69 ALDH1A1 (0.46) CYP1A2CYP3A4LMNAMAOAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832074-B1 AMINO ACID DERIVATIVES OF SUBSTITUTED QUINOXALINE 2,3-DIONE DERIVATIVES AS GLUTAMATE RECEPTOR ANTAGONISTS WARNER LAMBERT CO (US) 2002-09-04 EP disclosed
WO-1996040649-A1 AMINO ACID DERIVATIVES OF SUBSTITUTED QUINOXALINE 2,3-DIONE DERIVATIVES AS GLUTAMATE RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1996-12-19 WO disclosed