SCHEMBL7586348

SCHEMBL7586348

COc1ccc(C(=O)c2ccc(F)cc2Cl)cc1Cc1ccc(=O)[nH]n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 4/20 0.41
PLA2G2A P14555 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
NPC1 O15118 1/20 0.39
CYP3A4 P08684 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
PTGER1 P34995 2/20 0.38
ALDH1A1 P00352 2/20 0.38
GAA P10253 2/20 0.38
ROCK2 O75116 2/20 0.37
ROCK1 Q13464 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ADRB2 P07550 1/20 0.37
LMNA P02545 1/20 0.37
PKM P14618 1/20 0.37
AKR1B1 P15121 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7585660 0.84 ADRB2 (0.44) MAPTRAB9ACYP3A4ALDH1A1MEN1
SCHEMBL7584819 0.83 ADRB2 (0.39) MAPTCYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8502095 0.80 ROCK2 (0.39) PYGLPLA2G2AMAPTRAB9ANPC1
SCHEMBL7590521 0.80 HPGD (0.48) MAPTCYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL7583126 0.80 ADRB2 (0.39) MAPTCYP3A4ALDH1A1GAAADRB2
SCHEMBL7583504 0.77 ALDH1A1 (0.40) MAPTCYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL7583097 0.74 ALDH1A1 (0.41) MAPTRAB9ANPC1CYP3A4CYP1A2
SCHEMBL8502094 0.74 MEN1 (0.45) PYGLPLA2G2AMAPTPTGER1ALDH1A1
SCHEMBL7276846 0.74 PDE4A (0.45) MAPTCYP1A2CYP2C9CYP2C19GAA
Hydrochloric Acid SCHEMBL7274487 0.73 PDE4A (0.44) MAPTCYP1A2CYP2C9CYP2C19GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810218-B1 6-Benzyl-2H-pyridazin-3-one derivatives,their preparation and their use as inhibitors of prostaglandin G/H synthase I and II (COX I and COX II) HOFFMANN LA ROCHE (CH) 2002-12-04 EP disclosed
EP-0810218-A1 6-Benzyl-2H-pyridazin-3-one derivatives,their preparation and their use as inhibitors of prostaglandin G/H synthase I and II (COX I and COX II) F. HOFFMANN-LA ROCHE AG (CH) 1997-12-03 EP disclosed