SCHEMBL7587254

SCHEMBL7587254

CN(C)CC1=C(c2cccc(O)c2)c2ccc3ccccc3c2CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.41
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
NPY1R P25929 1/20 0.41
HTT P42858 1/20 0.41
NPY2R P49146 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
ATM Q13315 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36
MCL1 Q07820 1/20 0.35
LCK P06239 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7590974 0.83 HSD17B1 (0.36) ALDH1A1HSD17B1HSD17B2HTR7ESR2
Hydrochloric Acid SCHEMBL8011897 0.82 OPRK1 (0.35) ALDH1A1HSD17B1HSD17B2HTR7ESR2
SCHEMBL7605203 0.82 MAPT (0.39) MAPTALDH1A1NPC1LMNAHPGD
SCHEMBL7588577 0.82 HSD17B1 (0.35) HSD17B1HSD17B2ESR1ESR2
Hydrochloric Acid SCHEMBL8022870 0.81 MAPT (0.38) MAPTALDH1A1NPC1LMNAHPGD
Hydrochloric Acid SCHEMBL8014383 0.81 HSD17B1 (0.34) HSD17B1HSD17B2ESR1ESR2
SCHEMBL7584081 0.80 HSD17B1 (0.40) HSD17B1HSD17B2CYP1A2PIM1PIM2
Hydrochloric Acid SCHEMBL8017915 0.79 HSD17B1 (0.39) HSD17B1HSD17B2CYP1A2PIM1PIM2
SCHEMBL7591741 0.78 MTNR1A (0.44) MAPTALDH1A1LMNAKDM4EHSD17B1
SCHEMBL7588665 0.78 ESR1 (0.40) HSD17B1HSD17B2ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed