SCHEMBL7584081

SCHEMBL7584081

CN(C)CC1=C(c2cccc(O)c2)c2cc3ccccc3cc2CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 5/20 0.40
HSD17B2 P37059 5/20 0.40
GAPDH P04406 1/20 0.36
OPRK1 P41145 1/20 0.35
ESR1 P03372 4/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP2C19 P33261 1/20 0.35
ESR2 Q92731 1/20 0.35
PIK3CA P42336 1/20 0.34
OPRD1 P41143 3/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
PIM1 P11309 1/20 0.33
PIM2 Q9P1W9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8017915 0.99 HSD17B1 (0.39) HSD17B1HSD17B2GAPDHOPRK1ESR1
SCHEMBL27507099 0.87 MTNR1A (0.39) OPRK1ESR1CYP1A2CYP2D6ESR2
SCHEMBL7591741 0.86 MTNR1A (0.44) HSD17B1HSD17B2OPRK1CYP1A2CYP3A4
SCHEMBL7584146 0.86 PBRM1 (0.40) HSD17B1HSD17B2OPRK1ESR1CYP1A2
SCHEMBL7588665 0.86 ESR1 (0.40) HSD17B1HSD17B2ESR1ESR2CHRNB4
Hydrochloric Acid SCHEMBL8010759 0.85 MTNR1A (0.43) HSD17B1HSD17B2OPRK1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL8017505 0.85 PBRM1 (0.39) HSD17B1HSD17B2OPRK1ESR1CYP1A2
SCHEMBL7588071 0.85 TDP2 (0.41) HSD17B1HSD17B2OPRK1ESR1CYP1A2
Hydrochloric Acid SCHEMBL8017994 0.85 ESR1 (0.39) HSD17B1HSD17B2ESR1ESR2CHRNB4
SCHEMBL7585672 0.84 OPRK1 (0.46) HSD17B1HSD17B2OPRK1ESR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed