SCHEMBL7590192

SCHEMBL7590192

COc1ccc(Cc2c(C)cc(N3CCCC3)cc2C)cc1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
TSHR P16473 1/20 0.43
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
THRB P10828 9/20 0.39
THRA P10827 8/20 0.39
HIF1A Q16665 3/20 0.37
MAPT P10636 2/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
CHKA P35790 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
ALOX12 P18054 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7114452 0.80 THRB (0.50) THRBTHRAGAA
SCHEMBL666032 0.79 THRB (0.43) ALDH1A1THRBTHRAGAAALOX12
SCHEMBL6864460 0.79 THRB (0.48) ALDH1A1THRBTHRAMAPTKDM4E
SCHEMBL282445 0.79 THRB (0.49) THRBTHRAALOX12
SCHEMBL13913523 0.77 ALDH1A1 (0.54) ALDH1A1TSHRMEN1KMT2AHIF1A
SCHEMBL7555866 0.77 THRB (0.47) ALDH1A1TSHRMEN1KMT2ATHRB
SCHEMBL667473 0.77 THRB (0.45) ALDH1A1TSHRMEN1KMT2ATHRB
SCHEMBL7597002 0.76 THRB (0.47) ALDH1A1TSHRMEN1KMT2ATHRB
SCHEMBL667776 0.73 THRB (0.39) ALDH1A1THRBTHRAHIF1AMAPT
SCHEMBL6864242 0.73 THRB (0.49) THRBTHRAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194422-A1 BIARYL COMPOUNDS UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER (US) 2002-04-10 EP disclosed
WO-2000073292-A1 BIARYL COMPOUNDS THE UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER (US) 2000-12-07 WO disclosed