SCHEMBL7590256

SCHEMBL7590256

C[C@@H](CN(C)C)C(=O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
KDM4E B2RXH2 2/20 0.56
USP2 O75604 1/20 0.56
SMN1; SMN2 Q16637 7/20 0.54
HTT P42858 5/20 0.54
LMNA P02545 4/20 0.54
MAPT P10636 5/20 0.54
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
MAPK1 P28482 1/20 0.53
ATM Q13315 1/20 0.53
EGFR P00533 1/20 0.51
PDCD1 Q15116 1/20 0.47
CD274 Q9NZQ7 1/20 0.47
HPGD P15428 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7590251 1.00 ALDH1A1 (0.56) ALDH1A1KDM4EUSP2SMN1; SMN2HTT
SCHEMBL6726553 0.90 NPC1 (0.64) ALDH1A1HTTLMNAMAPTNPC1
SCHEMBL9683311 0.90 NPC1 (0.64) ALDH1A1HTTLMNAMAPTNPC1
Hydrochloric Acid SCHEMBL9324495 0.88 MAPT (0.67) ALDH1A1HTTLMNAMAPTNPC1
Hydrochloric Acid SCHEMBL10353456 0.86 EGFR (0.58) ALDH1A1SMN1; SMN2HTTLMNAMAPT
SCHEMBL11439856 0.83 EGFR (0.57) ALDH1A1SMN1; SMN2HTTLMNAMAPT
SCHEMBL9850638 0.81 CHRM2 (0.51) ALDH1A1KDM4ESMN1; SMN2HTTLMNA
SCHEMBL4558930 0.81 SMN1; SMN2 (0.56) ALDH1A1KDM4EUSP2SMN1; SMN2HTT
SCHEMBL9850647 0.79 EGFR (0.50) ALDH1A1KDM4ESMN1; SMN2HTTLMNA
SCHEMBL9859087 0.79 EGFR (0.50) ALDH1A1SMN1; SMN2HTTLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0864559-B1 Substituted amino compounds and their use as analgesic active substances GRUENENTHAL GMBH (DE) 2002-06-05 EP disclosed
US-6022895-A Substituted amino compounds and their use as substances having an analgesic effect GRUENENTHAL GMBH (DE) 2000-02-08 US disclosed
EP-0864559-A1 Substituted amino compounds and their use as analgesic active substances Grünenthal GmbH (DE) 1998-09-16 EP disclosed